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All rights reserved. http://resource.belframework.org/belframework/20131211/knowledge/large_corpus.bel http://purl.org/dc/elements/1.1/title BEL Framework Large Corpus Document http://resource.belframework.org/belframework/20131211/knowledge/large_corpus.bel http://purl.org/pav/authoredBy http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#_5 http://resource.belframework.org/belframework/20131211/knowledge/large_corpus.bel http://purl.org/pav/version 20131211 http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#_4 http://www.w3.org/ns/prov#value A class of high-affinity inhibitors is disclosed that selectively target and irreversibly inactivate the epidermal growth factor receptor tyrosine kinase through specific, covalent modification of a cysteine residue present in the ATP binding pocket. ..Evidence is also presented to indicate that the compounds interact in an analogous fashion with erbB2 but have no activity against the other receptor tyrosine kinases or intracellular tyrosine kinases that were tested in this study. http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#_4 http://www.w3.org/ns/prov#wasQuotedFrom http://www.ncbi.nlm.nih.gov/pubmed/9751783 http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#_5 http://www.w3.org/2000/01/rdf-schema#label Selventa http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#assertion http://www.w3.org/ns/prov#hadPrimarySource http://www.ncbi.nlm.nih.gov/pubmed/9751783 http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#assertion http://www.w3.org/ns/prov#wasDerivedFrom http://resource.belframework.org/belframework/20131211/knowledge/large_corpus.bel http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#assertion http://www.w3.org/ns/prov#wasDerivedFrom http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#_4 http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s#pubinfo http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s http://purl.org/dc/terms/created 2014-07-03T14:34:16.137+02:00 http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s http://purl.org/pav/createdBy http://orcid.org/0000-0001-6818-334X http://www.tkuhn.ch/bel2nanopub/RASisEF6XNvbUDo9FeD6fmRntcpsVFDrtA89KBON6fl1s http://purl.org/pav/createdBy http://orcid.org/0000-0002-1267-0234