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Transfection of AhRR expression vector into HeLa cells, together with the expression vectors of AhR and Arnt and the reporter gene pX4TK–Luc, repressed luciferase expression originally induced by AhR and Arnt plasmids in a dose-dependent fashion (Fig. 3A, lanes 3–5). This repression was reversed by further addition of AhR expression vector (data not shown). These results indicate that AhRR functions as a competitive repressor of AhR.
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